Temperature-Controlled Diastereoselective Doebner/Ugi Tandem Reaction
Novel peptidomimetics containing a pyrrolone fragment were synthesized by a tandem combination of Doebner and Ugi type multicomponent reactions with controlled diastereoselectivity. This approach represents a convenient synthesis in the temperature range from 25 to 45 °C. In most cases, the new method allowed each diastereomer to be isolated separately.
- Location
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Deutsche Nationalbibliothek Frankfurt am Main
- Extent
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Online-Ressource
- Language
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Englisch
- Bibliographic citation
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Temperature-Controlled Diastereoselective Doebner/Ugi Tandem Reaction ; volume:07 ; number:02 ; year:2023 ; pages:258-266
SynOpen ; 07, Heft 02 (2023), 258-266
- Contributor
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Sakhno, Yana
Radchenko, Oleksandr
Saraev, Vyacheslav
Shliapkina, Yuliia
Kaidash, Mariia
Shyshkina, Mariia
Shishkina, Svitlana
Musatov, Vladimir
Desenko, Sergey
Chebanov, Valentyn
- DOI
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10.1055/a-2091-7934
- URN
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urn:nbn:de:101:1-2023072010271213737547
- Rights
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Open Access; Der Zugriff auf das Objekt ist unbeschränkt möglich.
- Last update
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14.08.2025, 10:45 AM CEST
Data provider
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Associated
- Sakhno, Yana
- Radchenko, Oleksandr
- Saraev, Vyacheslav
- Shliapkina, Yuliia
- Kaidash, Mariia
- Shyshkina, Mariia
- Shishkina, Svitlana
- Musatov, Vladimir
- Desenko, Sergey
- Chebanov, Valentyn
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Ugi, Luise
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Diastereoselective Ugi reaction of chiral 1,3-aminoalcohols derived from an organocatalytic Mannich reaction
Novel postmodifications of the Ugi reaction
Unimolecular Exciplexes by Ugi Four-Component Reaction
Post-Ugi gold-catalyzed diastereoselective domino cyclization for the synthesis of diversely substituted spiroindolines
Cobalt-Catalyzed Enantio- and Diastereoselective Hydroacylation Reaction
Asymmetric Phosphoric Acid Catalyzed Four-Component Ugi Reaction
Site‐Selective Protein Conjugation by a Multicomponent Ugi Reaction
Synthesis of Sulfonyl Fluoro Peptides by an Ugi Reaction
Effective microwave-assisted approach to 1,2,3-triazolobenzodiazepinones via tandem Ugi reaction/catalyst-free intramolecular azide–alkyne cycloaddition
Ugi, Luise
Ugi, Oskar
Ugi, Ivar
Diastereoselective Ugi reaction of chiral 1,3-aminoalcohols derived from an organocatalytic Mannich reaction
Novel postmodifications of the Ugi reaction
Unimolecular Exciplexes by Ugi Four-Component Reaction
Post-Ugi gold-catalyzed diastereoselective domino cyclization for the synthesis of diversely substituted spiroindolines
Cobalt-Catalyzed Enantio- and Diastereoselective Hydroacylation Reaction
Asymmetric Phosphoric Acid Catalyzed Four-Component Ugi Reaction
Site‐Selective Protein Conjugation by a Multicomponent Ugi Reaction
Synthesis of Sulfonyl Fluoro Peptides by an Ugi Reaction
Effective microwave-assisted approach to 1,2,3-triazolobenzodiazepinones via tandem Ugi reaction/catalyst-free intramolecular azide–alkyne cycloaddition
Ugi, Luise
Ugi, Oskar