Temperature-Controlled Diastereoselective Doebner/Ugi Tandem Reaction
Novel peptidomimetics containing a pyrrolone fragment were synthesized by a tandem combination of Doebner and Ugi type multicomponent reactions with controlled diastereoselectivity. This approach represents a convenient synthesis in the temperature range from 25 to 45 °C. In most cases, the new method allowed each diastereomer to be isolated separately.
- Standort
-
Deutsche Nationalbibliothek Frankfurt am Main
- Umfang
-
Online-Ressource
- Sprache
-
Englisch
- Erschienen in
-
Temperature-Controlled Diastereoselective Doebner/Ugi Tandem Reaction ; volume:07 ; number:02 ; year:2023 ; pages:258-266
SynOpen ; 07, Heft 02 (2023), 258-266
- Beteiligte Personen und Organisationen
-
Sakhno, Yana
Radchenko, Oleksandr
Saraev, Vyacheslav
Shliapkina, Yuliia
Kaidash, Mariia
Shyshkina, Mariia
Shishkina, Svitlana
Musatov, Vladimir
Desenko, Sergey
Chebanov, Valentyn
- DOI
-
10.1055/a-2091-7934
- URN
-
urn:nbn:de:101:1-2023072010271213737547
- Rechteinformation
-
Open Access; Der Zugriff auf das Objekt ist unbeschränkt möglich.
- Letzte Aktualisierung
-
14.08.2025, 10:45 MESZ
Datenpartner
Dieses Objekt wird bereitgestellt von:
Deutsche Nationalbibliothek. Bei Fragen zum Objekt wenden Sie sich bitte an den Datenpartner.
Deutsche Nationalbibliothek. Bei Fragen zum Objekt wenden Sie sich bitte an den Datenpartner.
Beteiligte
- Sakhno, Yana
- Radchenko, Oleksandr
- Saraev, Vyacheslav
- Shliapkina, Yuliia
- Kaidash, Mariia
- Shyshkina, Mariia
- Shishkina, Svitlana
- Musatov, Vladimir
- Desenko, Sergey
- Chebanov, Valentyn
Ähnliche Objekte (12)
Diastereoselective Ugi reaction of chiral 1,3-aminoalcohols derived from an organocatalytic Mannich reaction
Novel postmodifications of the Ugi reaction
Cobalt-Catalyzed Enantio- and Diastereoselective Hydroacylation Reaction
Post-Ugi gold-catalyzed diastereoselective domino cyclization for the synthesis of diversely substituted spiroindolines
Unimolecular Exciplexes by Ugi Four-Component Reaction
Asymmetric Phosphoric Acid Catalyzed Four-Component Ugi Reaction
Site‐Selective Protein Conjugation by a Multicomponent Ugi Reaction
Synthesis of Sulfonyl Fluoro Peptides by an Ugi Reaction
Effective microwave-assisted approach to 1,2,3-triazolobenzodiazepinones via tandem Ugi reaction/catalyst-free intramolecular azide–alkyne cycloaddition
Synthesis of Sterically Hindered Tripeptides Using a Modified Ugi Reaction
Protein‐Templated Hit Identification through an Ugi Four‐Component Reaction **
Ugi, Ivar
Diastereoselective Ugi reaction of chiral 1,3-aminoalcohols derived from an organocatalytic Mannich reaction
Novel postmodifications of the Ugi reaction
Cobalt-Catalyzed Enantio- and Diastereoselective Hydroacylation Reaction
Post-Ugi gold-catalyzed diastereoselective domino cyclization for the synthesis of diversely substituted spiroindolines
Unimolecular Exciplexes by Ugi Four-Component Reaction
Asymmetric Phosphoric Acid Catalyzed Four-Component Ugi Reaction
Site‐Selective Protein Conjugation by a Multicomponent Ugi Reaction
Synthesis of Sulfonyl Fluoro Peptides by an Ugi Reaction
Effective microwave-assisted approach to 1,2,3-triazolobenzodiazepinones via tandem Ugi reaction/catalyst-free intramolecular azide–alkyne cycloaddition
Synthesis of Sterically Hindered Tripeptides Using a Modified Ugi Reaction
Protein‐Templated Hit Identification through an Ugi Four‐Component Reaction **
Ugi, Ivar
Diastereoselective Ugi reaction of chiral 1,3-aminoalcohols derived from an organocatalytic Mannich reaction
Novel postmodifications of the Ugi reaction
Cobalt-Catalyzed Enantio- and Diastereoselective Hydroacylation Reaction
Post-Ugi gold-catalyzed diastereoselective domino cyclization for the synthesis of diversely substituted spiroindolines
Unimolecular Exciplexes by Ugi Four-Component Reaction
Asymmetric Phosphoric Acid Catalyzed Four-Component Ugi Reaction
Site‐Selective Protein Conjugation by a Multicomponent Ugi Reaction
Synthesis of Sulfonyl Fluoro Peptides by an Ugi Reaction
Effective microwave-assisted approach to 1,2,3-triazolobenzodiazepinones via tandem Ugi reaction/catalyst-free intramolecular azide–alkyne cycloaddition
Synthesis of Sterically Hindered Tripeptides Using a Modified Ugi Reaction
Protein‐Templated Hit Identification through an Ugi Four‐Component Reaction **