Synthesis of novel glycosyl 1,3,4-oxadiazole derivatives

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Abstract: A convenient and practical protocol was developed to synthesize glycosyl 1,3,4-oxadiazoles from d-glucosamine with good to excellent yields. The key step involved p-TsCl/pyridine-mediated cyclization under mild conditions. Subsequent removal of the acetyl groups in the last step, conducted using the system of NaOMe/MeOH, gave the desired N-acetyl-d-glucosamine 1,3,4-oxadiazole derivatives.

Location: Deutsche Nationalbibliothek Frankfurt am Main

Extent: Online-Ressource

Language: Englisch

Bibliographic citation: Synthesis of novel glycosyl 1,3,4-oxadiazole derivatives ; volume:20 ; number:6 ; year:2014 ; pages:333-338 ; extent:6
Heterocyclic communications ; 20, Heft 6 (2014), 333-338 (gesamt 6)

Creator: Liu, Weiwei
Li, Quxiang
Cheng, Fengchang
Shi, Dahua
Cao, Zhiling

DOI: 10.1515/hc-2014-0166

URN: urn:nbn:de:101:1-2501130542508.923500918357

Rights: Open Access; Der Zugriff auf das Objekt ist unbeschränkt möglich.

Last update: 15.08.2025, 7:39 AM CEST

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Liu, Weiwei
Li, Quxiang
Cheng, Fengchang
Shi, Dahua
Cao, Zhiling

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Synthesis of novel glycosyl 1,3,4-oxadiazole derivatives

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Other Objects (12)

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