Synthesis of novel glycosyl 1,3,4-oxadiazole derivatives
Abstract: A convenient and practical protocol was developed to synthesize glycosyl 1,3,4-oxadiazoles from d-glucosamine with good to excellent yields. The key step involved p-TsCl/pyridine-mediated cyclization under mild conditions. Subsequent removal of the acetyl groups in the last step, conducted using the system of NaOMe/MeOH, gave the desired N-acetyl-d-glucosamine 1,3,4-oxadiazole derivatives.
- Standort
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Deutsche Nationalbibliothek Frankfurt am Main
- Umfang
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Online-Ressource
- Sprache
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Englisch
- Erschienen in
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Synthesis of novel glycosyl 1,3,4-oxadiazole derivatives ; volume:20 ; number:6 ; year:2014 ; pages:333-338 ; extent:6
Heterocyclic communications ; 20, Heft 6 (2014), 333-338 (gesamt 6)
- Urheber
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Liu, Weiwei
Li, Quxiang
Cheng, Fengchang
Shi, Dahua
Cao, Zhiling
- DOI
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10.1515/hc-2014-0166
- URN
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urn:nbn:de:101:1-2501130542508.923500918357
- Rechteinformation
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Open Access; Der Zugriff auf das Objekt ist unbeschränkt möglich.
- Letzte Aktualisierung
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15.08.2025, 07:39 MESZ
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Beteiligte
- Liu, Weiwei
- Li, Quxiang
- Cheng, Fengchang
- Shi, Dahua
- Cao, Zhiling
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