Synthesis of H4 pantetheine adducts for histone acetyltransferase inhibition
Abstract: Site-specific modifications of peptides provide a powerful tool for design of chemical probes and enzyme inhibitors. A convenient synthesis method was developed and used to produce H4K16-pantetheine bisubstrate analogs which could be employed as inhibitors of histone acetyltransferases in vivo and in vitro.
- Location
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Deutsche Nationalbibliothek Frankfurt am Main
- Extent
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Online-Ressource
- Language
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Englisch
- Bibliographic citation
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Synthesis of H4 pantetheine adducts for histone acetyltransferase inhibition ; volume:16 ; number:4-6 ; year:2010 ; pages:231-234
Heterocyclic communications ; 16, Heft 4-6 (2010), 231-234
- Creator
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Wu, Jiang
Zheng, Yujun George
- DOI
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10.1515/HC.2010.014
- URN
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urn:nbn:de:101:1-2501130541512.734231721710
- Rights
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Open Access; Der Zugriff auf das Objekt ist unbeschränkt möglich.
- Last update
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15.08.2025, 7:24 AM CEST
Data provider
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Associated
- Wu, Jiang
- Zheng, Yujun George
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