Phenol‐benzoxazolone bioisosteres of GluN2B‐NMDA receptor antagonists: Unexpected rearrangement during reductive alkylation with phenylcyclohexanone

to related objects

Location: Deutsche Nationalbibliothek Frankfurt am Main

Extent: Online-Ressource

Language: Englisch

Bibliographic citation: Phenol‐benzoxazolone bioisosteres of GluN2B‐NMDA receptor antagonists: Unexpected rearrangement during reductive alkylation with phenylcyclohexanone ; day:30 ; month:07 ; year:2022 ; extent:11
Archiv der Pharmazie ; (30.07.2022) (gesamt 11)

Creator: Markus, Alexander
Schreiber, Julian A.
Goerges, Gunnar
Frehland, Bastian
Schepmann, Dirk
Daniliuc, Constantin Gabriel
Fröhlich, Roland
Seebohm, Guiscard
Wünsch, Bernhard

DOI: 10.1002/ardp.202200225

URN: urn:nbn:de:101:1-2022073115050645760804

Rights: Open Access; Der Zugriff auf das Objekt ist unbeschränkt möglich.

Last update: 15.08.2025, 7:25 AM CEST

Data provider

This object is provided by:
Deutsche Nationalbibliothek. If you have any questions about the object, please contact the data provider.

Show original at data provider

Associated

Markus, Alexander
Schreiber, Julian A.
Goerges, Gunnar
Frehland, Bastian
Schepmann, Dirk
Daniliuc, Constantin Gabriel
Fröhlich, Roland
Seebohm, Guiscard
Wünsch, Bernhard

Other Objects (12)

Quinolone bioisosteres of phenolic GluN2B‐selective NMDA receptor antagonists

Hochschulschrift

GluN2B selective NMDA receptor antagonists : design, synthesis, pharmacological evaluation and docking studies

[2.2]Paracyclophane‐Based TCN‐201 Analogs as GluN2A‐Selective NMDA Receptor Antagonists

Unmasking GluN1/GluN3A excitatory glycine NMDA receptors

Indium-Catalyzed Reductive Alkylation of Indoles

Positive Modulatory Interactions of NMDA Receptor GluN1/2B Ligand Binding Domains Attenuate Antagonists Activity

Aufsatzsammlung

NMDA antagonists as potential analgesic drugs

Hochschulschrift

Synthesis and biological evaluation of ß-and y-amino alcohols as GluN2B selective NMDA receptor antagonists

Hochschulschrift

Characterization of NMDA receptors and investigation of the influence of GluN2B antagonists in pancreatic islet-cells

GluN2A‐Selective NMDA Receptor Antagonists: Mimicking the U‐Shaped Bioactive Conformation of TCN‐201 by a (2.2) Paracyclophane System

Hochschulschrift

Untersuchungen zu molekularen Interaktions- und Inhibitionsmechanismen von GluN2A- und GluN2B-selektiven NMDA-Rezeptorantagonisten

Brain networks in pharmacological fMRI of NMDA antagonists

Quinolone bioisosteres of phenolic GluN2B‐selective NMDA receptor antagonists

Hochschulschrift

GluN2B selective NMDA receptor antagonists : design, synthesis, pharmacological evaluation and docking studies

[2.2]Paracyclophane‐Based TCN‐201 Analogs as GluN2A‐Selective NMDA Receptor Antagonists

Unmasking GluN1/GluN3A excitatory glycine NMDA receptors

Indium-Catalyzed Reductive Alkylation of Indoles

Positive Modulatory Interactions of NMDA Receptor GluN1/2B Ligand Binding Domains Attenuate Antagonists Activity

Aufsatzsammlung

NMDA antagonists as potential analgesic drugs

Hochschulschrift

Synthesis and biological evaluation of ß-and y-amino alcohols as GluN2B selective NMDA receptor antagonists

Hochschulschrift

Characterization of NMDA receptors and investigation of the influence of GluN2B antagonists in pancreatic islet-cells

GluN2A‐Selective NMDA Receptor Antagonists: Mimicking the U‐Shaped Bioactive Conformation of TCN‐201 by a (2.2) Paracyclophane System

Hochschulschrift

Untersuchungen zu molekularen Interaktions- und Inhibitionsmechanismen von GluN2A- und GluN2B-selektiven NMDA-Rezeptorantagonisten

Brain networks in pharmacological fMRI of NMDA antagonists

Quinolone bioisosteres of phenolic GluN2B‐selective NMDA receptor antagonists

Hochschulschrift

GluN2B selective NMDA receptor antagonists : design, synthesis, pharmacological evaluation and docking studies

[2.2]Paracyclophane‐Based TCN‐201 Analogs as GluN2A‐Selective NMDA Receptor Antagonists

Unmasking GluN1/GluN3A excitatory glycine NMDA receptors

Indium-Catalyzed Reductive Alkylation of Indoles

Positive Modulatory Interactions of NMDA Receptor GluN1/2B Ligand Binding Domains Attenuate Antagonists Activity

Aufsatzsammlung

NMDA antagonists as potential analgesic drugs

Hochschulschrift

Synthesis and biological evaluation of ß-and y-amino alcohols as GluN2B selective NMDA receptor antagonists

Hochschulschrift

Characterization of NMDA receptors and investigation of the influence of GluN2B antagonists in pancreatic islet-cells

GluN2A‐Selective NMDA Receptor Antagonists: Mimicking the U‐Shaped Bioactive Conformation of TCN‐201 by a (2.2) Paracyclophane System

Hochschulschrift

Untersuchungen zu molekularen Interaktions- und Inhibitionsmechanismen von GluN2A- und GluN2B-selektiven NMDA-Rezeptorantagonisten

Brain networks in pharmacological fMRI of NMDA antagonists

Cultural heritage institutions wishing to register will find more information here.

Fields marked * need to be filled in.

Username*

Please enter your username

Email*

Please enter your email address

Please do not fill this field

First name

Last name

Password*

Please enter your password

Confirm password*

Please enter the same password

I have read the terms of use and the privacy policy for the collection of personal data and accept them. *

This field is required.

I would like to subscribe to the newsletter of the Deutsche Digitale Bibliothek. See newsletter subscription info.

Account created

Your "My DDB" account has been successfully created. Before you can log in to your account, you must click the confirmation link in the message we just sent to the email address you provided.

Phenol‐benzoxazolone bioisosteres of GluN2B‐NMDA receptor antagonists: Unexpected rearrangement during reductive alkylation with phenylcyclohexanone

Object Details

References and Relationships

Contributors, Places and Time

Further information

Data provider

Associated

Other Objects (12)

Quinolone bioisosteres of phenolic GluN2B‐selective NMDA receptor antagonists

GluN2B selective NMDA receptor antagonists : design, synthesis, pharmacological evaluation and docking studies

[2.2]Paracyclophane‐Based TCN‐201 Analogs as GluN2A‐Selective NMDA Receptor Antagonists

Unmasking GluN1/GluN3A excitatory glycine NMDA receptors

Indium-Catalyzed Reductive Alkylation of Indoles

Positive Modulatory Interactions of NMDA Receptor GluN1/2B Ligand Binding Domains Attenuate Antagonists Activity

NMDA antagonists as potential analgesic drugs

Synthesis and biological evaluation of ß-and y-amino alcohols as GluN2B selective NMDA receptor antagonists

Characterization of NMDA receptors and investigation of the influence of GluN2B antagonists in pancreatic islet-cells

GluN2A‐Selective NMDA Receptor Antagonists: Mimicking the U‐Shaped Bioactive Conformation of TCN‐201 by a (2.2) Paracyclophane System

Untersuchungen zu molekularen Interaktions- und Inhibitionsmechanismen von GluN2A- und GluN2B-selektiven NMDA-Rezeptorantagonisten

Brain networks in pharmacological fMRI of NMDA antagonists

Quinolone bioisosteres of phenolic GluN2B‐selective NMDA receptor antagonists

GluN2B selective NMDA receptor antagonists : design, synthesis, pharmacological evaluation and docking studies

[2.2]Paracyclophane‐Based TCN‐201 Analogs as GluN2A‐Selective NMDA Receptor Antagonists

Unmasking GluN1/GluN3A excitatory glycine NMDA receptors

Indium-Catalyzed Reductive Alkylation of Indoles

Positive Modulatory Interactions of NMDA Receptor GluN1/2B Ligand Binding Domains Attenuate Antagonists Activity

NMDA antagonists as potential analgesic drugs

Synthesis and biological evaluation of ß-and y-amino alcohols as GluN2B selective NMDA receptor antagonists

Characterization of NMDA receptors and investigation of the influence of GluN2B antagonists in pancreatic islet-cells

GluN2A‐Selective NMDA Receptor Antagonists: Mimicking the U‐Shaped Bioactive Conformation of TCN‐201 by a (2.2) Paracyclophane System

Untersuchungen zu molekularen Interaktions- und Inhibitionsmechanismen von GluN2A- und GluN2B-selektiven NMDA-Rezeptorantagonisten

Brain networks in pharmacological fMRI of NMDA antagonists

Quinolone bioisosteres of phenolic GluN2B‐selective NMDA receptor antagonists

GluN2B selective NMDA receptor antagonists : design, synthesis, pharmacological evaluation and docking studies

[2.2]Paracyclophane‐Based TCN‐201 Analogs as GluN2A‐Selective NMDA Receptor Antagonists

Unmasking GluN1/GluN3A excitatory glycine NMDA receptors

Indium-Catalyzed Reductive Alkylation of Indoles

Positive Modulatory Interactions of NMDA Receptor GluN1/2B Ligand Binding Domains Attenuate Antagonists Activity

NMDA antagonists as potential analgesic drugs

Synthesis and biological evaluation of ß-and y-amino alcohols as GluN2B selective NMDA receptor antagonists

Characterization of NMDA receptors and investigation of the influence of GluN2B antagonists in pancreatic islet-cells

GluN2A‐Selective NMDA Receptor Antagonists: Mimicking the U‐Shaped Bioactive Conformation of TCN‐201 by a (2.2) Paracyclophane System

Untersuchungen zu molekularen Interaktions- und Inhibitionsmechanismen von GluN2A- und GluN2B-selektiven NMDA-Rezeptorantagonisten

Brain networks in pharmacological fMRI of NMDA antagonists

Related objects

Reset password