Synthesis of functionalized bicyclic pyridones containing the dithiocarbamate group using thioazlactones, diamines, and nitroketene dithioacetal

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Abstract: An efficient method for the synthesis of highly substituted bicyclic pyridone derivatives containing the dithiocarbamate group is reported via a one-pot three-component reaction of 2-(alkylthio)thioazlactones, diamines, and nitroketene dithioacetal in EtOH under catalyst-free conditions. The reaction proceeds via a domino amidation–intramolecular 1,4-addition-type Friedel–Crafts alkylation reaction to afford the corresponding fused bicyclic pyridones with high yields and diastereoselectivity

Location: Deutsche Nationalbibliothek Frankfurt am Main

Extent: Online-Ressource

Language: Englisch

Notes: SynOpen. - 05, 02 (2021) , 108-113, ISSN: 2509-9396

Event: Veröffentlichung

(where): Freiburg

(who): Universität

(when): 2024

Creator: Saeedi, Marziyeh
Khoshdoun, Maryam
Taheri, Salman
Ziyaei Halimehjani, Azim
Mohammadi, Aliasghar
Halvagar, Mohammad Reza
Amani, Vahid

DOI: 10.1055/a-1492-9229

URN: urn:nbn:de:bsz:25-freidok-2477218

Rights: Open Access; Der Zugriff auf das Objekt ist unbeschränkt möglich.

Last update: 14.08.2025, 10:59 AM CEST

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Associated

Saeedi, Marziyeh
Khoshdoun, Maryam
Taheri, Salman
Ziyaei Halimehjani, Azim
Mohammadi, Aliasghar
Halvagar, Mohammad Reza
Amani, Vahid
Universität

Time of origin

2024

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