Synthesis of (6,5,5) Ring‐Fused Tricyclic Triazoles by Copper‐Promoted Double Cyclization
Abstract: Ring‐fused 1,2,3‐triazoles are important biologically active compounds and synthetic intermediates. Known methods for their synthesis are limited mostly to triazoles fused to six‐membered or larger rings. Herein we disclose a synthetic approach to triazoles fused to five‐membered rings based on copper (I)‐promoted double cyclization consisting of azide‐alkyne cycloaddition, followed by cross coupling to aryl iodides.
- Standort
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Deutsche Nationalbibliothek Frankfurt am Main
- Umfang
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Online-Ressource
- Sprache
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Englisch
- Erschienen in
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Synthesis of (6,5,5) Ring‐Fused Tricyclic Triazoles by Copper‐Promoted Double Cyclization ; day:25 ; month:10 ; year:2024 ; extent:5
European journal of organic chemistry ; (25.10.2024) (gesamt 5)
- Urheber
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Pošta, Martin
Dmitrieva, Margarita
Volpe, Chiara
Matoušek, Václav
Klepetářová, Blanka
Beier, Petr
- DOI
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10.1002/ejoc.202400736
- URN
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urn:nbn:de:101:1-2410261428231.489653269176
- Rechteinformation
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Open Access; Der Zugriff auf das Objekt ist unbeschränkt möglich.
- Letzte Aktualisierung
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15.08.2025, 07:31 MESZ
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Beteiligte
- Pošta, Martin
- Dmitrieva, Margarita
- Volpe, Chiara
- Matoušek, Václav
- Klepetářová, Blanka
- Beier, Petr
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