A2A adenosine receptor antagonists: are triazolotriazine and purine scaffolds interchangeable?

to connected objects

Location: Deutsche Nationalbibliothek Frankfurt am Main

Extent: Online-Ressource

Language: Englisch

Bibliographic citation: In: Molecules (2022) 27:8, 2386. https://doi.org/10.3390/molecules27082386

Event: Veröffentlichung

(where): Würzburg

(who): Universität Würzburg

(when): 2023

Creator: Spinaci, Andrea
Lambertucci, Catia
Buccioni, Michela
Dal Ben, Diego
Graiff, Claudia
Barbalace, Maria Cristina
Hrelia, Silvana
Angeloni, Cristina
Tayebati, Seyed Khosrow
Ubaldi, Massimo
Masi, Alessio
Klotz, Karl-Norbert
Volpini, Rosaria
Marucci, Gabriella

DOI: 10.3390/molecules27082386

URN: urn:nbn:de:bvb:20-opus-270618

Rights: Der Zugriff auf das Objekt ist unbeschränkt möglich.

Last update: 25.03.2025, 1:51 PM CET

Data provider

This object is provided by:
Deutsche Nationalbibliothek. If you have any questions about the object, please contact the data provider.

Show original at data provider

Associated

Spinaci, Andrea
Lambertucci, Catia
Buccioni, Michela
Dal Ben, Diego
Graiff, Claudia
Barbalace, Maria Cristina
Hrelia, Silvana
Angeloni, Cristina
Tayebati, Seyed Khosrow
Ubaldi, Massimo
Masi, Alessio
Klotz, Karl-Norbert
Volpini, Rosaria
Marucci, Gabriella
Universität Würzburg

Time of origin

2023

Other Objects (12)

Irreversible Antagonists for the Adenosine A2B Receptor

Barbiturates are selective antagonists at A1 adenosine receptors

8-Substituted 1,3-dimethyltetrahydropyrazino[2,1-f]purinediones: water-soluble adenosine receptor antagonists and monoamine oxidase B inhibitors

Hochschulschrift

Adenosine 2a receptor signaling in autoimmune neuroinflammation

Adenosine receptor agonists: Synthesis and biological evaluation of 1-deaza analogues of adenosine

Hochschulschrift

In vivo pharmacological profiling in Xenopus embryos defines a subset of A1 adenosine receptor-selective antagonists with potent anti-angiogenic activities

Multivalently binding antagonists for the neurokinin-1 receptor

Mechanism of A2 adenosine receptor activation. I. Blockade of A2 adenosine receptors by photoaffinity labeling

Histamine H3 receptor antagonists in combination with monoamine oxidase B and adenosine A1/A2A receptor ligands as multi-target approach for the treatment of Parkinson´s disease

Anticonvulsant effects of isomeric nonimidazole histamine H3 receptor antagonists

Structure-Based Development of Selective Orexin 1 Receptor Antagonists

Konferenzschrift | Kongress

The effects of beta receptor antagonists on the myorcardium

Irreversible Antagonists for the Adenosine A2B Receptor

Barbiturates are selective antagonists at A1 adenosine receptors

8-Substituted 1,3-dimethyltetrahydropyrazino[2,1-f]purinediones: water-soluble adenosine receptor antagonists and monoamine oxidase B inhibitors

Hochschulschrift

Adenosine 2a receptor signaling in autoimmune neuroinflammation

Adenosine receptor agonists: Synthesis and biological evaluation of 1-deaza analogues of adenosine

Hochschulschrift

In vivo pharmacological profiling in Xenopus embryos defines a subset of A1 adenosine receptor-selective antagonists with potent anti-angiogenic activities

Multivalently binding antagonists for the neurokinin-1 receptor

Mechanism of A2 adenosine receptor activation. I. Blockade of A2 adenosine receptors by photoaffinity labeling

Histamine H3 receptor antagonists in combination with monoamine oxidase B and adenosine A1/A2A receptor ligands as multi-target approach for the treatment of Parkinson´s disease

Anticonvulsant effects of isomeric nonimidazole histamine H3 receptor antagonists

Structure-Based Development of Selective Orexin 1 Receptor Antagonists

Konferenzschrift | Kongress

The effects of beta receptor antagonists on the myorcardium

Irreversible Antagonists for the Adenosine A2B Receptor

Barbiturates are selective antagonists at A1 adenosine receptors

8-Substituted 1,3-dimethyltetrahydropyrazino[2,1-f]purinediones: water-soluble adenosine receptor antagonists and monoamine oxidase B inhibitors

Hochschulschrift

Adenosine 2a receptor signaling in autoimmune neuroinflammation

Adenosine receptor agonists: Synthesis and biological evaluation of 1-deaza analogues of adenosine

Hochschulschrift

In vivo pharmacological profiling in Xenopus embryos defines a subset of A1 adenosine receptor-selective antagonists with potent anti-angiogenic activities

Multivalently binding antagonists for the neurokinin-1 receptor

Mechanism of A2 adenosine receptor activation. I. Blockade of A2 adenosine receptors by photoaffinity labeling

Histamine H3 receptor antagonists in combination with monoamine oxidase B and adenosine A1/A2A receptor ligands as multi-target approach for the treatment of Parkinson´s disease

Anticonvulsant effects of isomeric nonimidazole histamine H3 receptor antagonists

Structure-Based Development of Selective Orexin 1 Receptor Antagonists

Konferenzschrift | Kongress

The effects of beta receptor antagonists on the myorcardium

Cultural heritage institutions wishing to register will find more information here.

Fields marked * need to be filled in.

Username*

Please enter your username

Email*

Please enter your email address

Please do not fill this field

First name

Last name

Password*

Please enter your password

Confirm password*

Please enter the same password

I have read the terms of use and the privacy policy for the collection of personal data and accept them. *

This field is required.

I would like to subscribe to the newsletter of the Deutsche Digitale Bibliothek. See newsletter subscription info.

Account created

Your "My DDB" account has been successfully created. Before you can log in to your account, you must click the confirmation link in the message we just sent to the email address you provided.

A2A adenosine receptor antagonists: are triazolotriazine and purine scaffolds interchangeable?

Object Details

References and Relationships

Contributors, Places and Time

Further information

Data provider

Associated

Time of origin

Other Objects (12)

Irreversible Antagonists for the Adenosine A2B Receptor

Barbiturates are selective antagonists at A1 adenosine receptors

8-Substituted 1,3-dimethyltetrahydropyrazino[2,1-f]purinediones: water-soluble adenosine receptor antagonists and monoamine oxidase B inhibitors

Adenosine 2a receptor signaling in autoimmune neuroinflammation

Adenosine receptor agonists: Synthesis and biological evaluation of 1-deaza analogues of adenosine

In vivo pharmacological profiling in Xenopus embryos defines a subset of A1 adenosine receptor-selective antagonists with potent anti-angiogenic activities

Multivalently binding antagonists for the neurokinin-1 receptor

Mechanism of A2 adenosine receptor activation. I. Blockade of A2 adenosine receptors by photoaffinity labeling

Histamine H3 receptor antagonists in combination with monoamine oxidase B and adenosine A1/A2A receptor ligands as multi-target approach for the treatment of Parkinson´s disease

Anticonvulsant effects of isomeric nonimidazole histamine H3 receptor antagonists

Structure-Based Development of Selective Orexin 1 Receptor Antagonists

The effects of beta receptor antagonists on the myorcardium

Irreversible Antagonists for the Adenosine A2B Receptor

Barbiturates are selective antagonists at A1 adenosine receptors

8-Substituted 1,3-dimethyltetrahydropyrazino[2,1-f]purinediones: water-soluble adenosine receptor antagonists and monoamine oxidase B inhibitors

Adenosine 2a receptor signaling in autoimmune neuroinflammation

Adenosine receptor agonists: Synthesis and biological evaluation of 1-deaza analogues of adenosine

In vivo pharmacological profiling in Xenopus embryos defines a subset of A1 adenosine receptor-selective antagonists with potent anti-angiogenic activities

Multivalently binding antagonists for the neurokinin-1 receptor

Mechanism of A2 adenosine receptor activation. I. Blockade of A2 adenosine receptors by photoaffinity labeling

Histamine H3 receptor antagonists in combination with monoamine oxidase B and adenosine A1/A2A receptor ligands as multi-target approach for the treatment of Parkinson´s disease

Anticonvulsant effects of isomeric nonimidazole histamine H3 receptor antagonists

Structure-Based Development of Selective Orexin 1 Receptor Antagonists

The effects of beta receptor antagonists on the myorcardium

Irreversible Antagonists for the Adenosine A2B Receptor

Barbiturates are selective antagonists at A1 adenosine receptors

8-Substituted 1,3-dimethyltetrahydropyrazino[2,1-f]purinediones: water-soluble adenosine receptor antagonists and monoamine oxidase B inhibitors

Adenosine 2a receptor signaling in autoimmune neuroinflammation

Adenosine receptor agonists: Synthesis and biological evaluation of 1-deaza analogues of adenosine

In vivo pharmacological profiling in Xenopus embryos defines a subset of A1 adenosine receptor-selective antagonists with potent anti-angiogenic activities

Multivalently binding antagonists for the neurokinin-1 receptor

Mechanism of A2 adenosine receptor activation. I. Blockade of A2 adenosine receptors by photoaffinity labeling

Histamine H3 receptor antagonists in combination with monoamine oxidase B and adenosine A1/A2A receptor ligands as multi-target approach for the treatment of Parkinson´s disease

Anticonvulsant effects of isomeric nonimidazole histamine H3 receptor antagonists

Structure-Based Development of Selective Orexin 1 Receptor Antagonists

The effects of beta receptor antagonists on the myorcardium

Related objects

Reset password