One-Pot Synthesis of Diaryl Sulfonamides using an Iron- and Copper-Catalyzed Aryl C–H Amidation Process

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A one-pot, two-stage synthesis of diaryl sulfonamides using sequential iron and copper catalysis is developed. Regioselective para-iodination of activated arenes by the super Lewis acid, iron triflimide and N-iodosuccinimide (NIS), is followed by a copper (I)-catalyzed N-arylation reaction. The process is found to be applicable for the coupling of a range of anisoles, anilines and acetanilides with primary sulfonamides and is used for the one-pot synthesis of biologically important compounds.

Location: Deutsche Nationalbibliothek Frankfurt am Main

Extent: Online-Ressource

Language: Englisch

Bibliographic citation: One-Pot Synthesis of Diaryl Sulfonamides using an Iron- and Copper-Catalyzed Aryl C–H Amidation Process ; volume:54 ; number:20 ; year:2022 ; pages:4551-4560
Synthesis ; 54, Heft 20 (2022), 4551-4560

Contributor: Waddell, Lachlan J. N.
Henry, Martyn C.
Mostafa, Mohamed A. B.
Sutherland, Andrew

DOI: 10.1055/a-1884-6988

URN: urn:nbn:de:101:1-2022120811290733503243

Rights: Kein Open Access; Der Zugriff auf das Objekt ist unbeschränkt möglich.

Last update: 15.08.2025, 7:35 AM CEST

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Waddell, Lachlan J. N.
Henry, Martyn C.
Mostafa, Mohamed A. B.
Sutherland, Andrew

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One-Pot Synthesis of Diaryl Sulfonamides using an Iron- and Copper-Catalyzed Aryl C–H Amidation Process

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Other Objects (12)

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